CUMYL-THPINACA
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Chemical compound
Pharmaceutical compound
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| Formula | C23H27N3O2 |
| Molar mass | 377.488 g·mol−1 |
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CUMYL-THPINACA (also known as SGT-42) is an indazole-3-carboxamide based synthetic cannabinoid.[1] [2] CUMYL-THPINACA acts as a potent agonist for the cannabinoid receptors, with approximately 6x selectivity for CB1, having an EC50 of 0.1nM for human CB1 receptors and 0.59nM for human CB2 receptors.[3]
Legal status
[edit ]Sweden's public health agency suggested to classify CUMYL-THPINACA as hazardous substance on November 10, 2014.[4]
As of October 2015 CUMYL-THPINACA is a controlled substance in China.[5]
See also
[edit ]- 5F-CUMYL-PINACA
- 5F-SDB-006
- ADAMANTYL-THPINACA
- CUMYL-4CN-BINACA
- CUMYL-CBMINACA
- CUMYL-PICA
- CUMYL-PINACA
- SDB-006
- NNE1
References
[edit ]- ^ "CUMYL-THPINACA". Cayman Chemical. Retrieved 11 July 2015.
- ^ Monti MC, Scheurer E, Mercer-Chalmers-Bender K (July 2021). "Phase I In Vitro Metabolic Profiling of the Synthetic Cannabinoid Receptor Agonists CUMYL-THPINACA and ADAMANTYL-THPINACA". Metabolites. 11 (8): 470. doi:10.3390/metabo11080470 . PMC 8398790 . PMID 34436411.
- ^ WO 2014167530, Bowden MJ, Williamson JP, "Cannabinoid compounds", published 2014年10月16日
- ^ "Cannabinoider föreslås bli klassade som hälsofarlig vara" . Retrieved 11 July 2015.
- ^ "关于印发《非药用类麻醉药品和精神药品列管办法》的通知" (in Chinese). China Food and Drug Administration. 27 September 2015. Archived from the original on 1 October 2015. Retrieved 1 October 2015.
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