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Schema
>
Reaction
>
Entries
KIT mutants bind ripretinib
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authored
[InstanceEdit:9681395] Rothfels, Karen, 2020年04月01日
category
binding
compartment
[Compartment:876] plasma membrane
[Compartment:70101] cytosol
created
[InstanceEdit:9681381] Rothfels, Karen, 2020年04月01日
crossReference
[DatabaseIdentifier:11944977] Mondo:0011719
[DatabaseIdentifier:11944892] Mondo:0004992
dbId
9681382
disease
[Disease:1500689] cancer
[Disease:9661830] gastrointestinal stromal tumor
displayName
KIT mutants bind ripretinib
edited
[InstanceEdit:9686618] Rothfels, Karen, 2020年05月04日
entityFunctionalStatus
[EntityFunctionalStatus:9686617] gain_of_function of ripretinib-sensitive KIT mutants [plasma membrane]
eventOf
[Pathway:R-HSA-9669921] KIT mutants bind TKIs - Homo sapiens
input
[ChemicalDrug:R-ALL-9674322] ripretinib [cytosol]
[CandidateSet:R-HSA-9681384] ripretinib-sensitive KIT mutants [plasma membrane]
isChimeric
false
isInDisease
true
isInferred
false
literatureReference
[LiteratureReference:9674274] Ripretinib (DCC-2618) Is a Switch Control Kinase Inhibitor of a Broad Spectrum of Oncogenic and Drug-Resistant KIT and PDGFRA Variants
[LiteratureReference:9727098] New drugs in gastrointestinal stromal tumors
maxDepth
1
modified
[InstanceEdit:9830342] Matthews, Lisa, 2023年03月08日
name
KIT mutants bind ripretinib
normalReaction
[Reaction:R-HSA-9681375] KIT binds ripretinib
output
[Complex:R-HSA-9681383] ripretinib-sensitive KIT:ripretinib [plasma membrane]
releaseDate
2020年06月10日
reviewStatus
[ReviewStatus:9821382] five stars
reviewed
[InstanceEdit:9678239] Serrano, C駸ar, 2020年03月13日
[InstanceEdit:9678232] Garc?a-Valverde, Alfonso, 2020年03月13日
[InstanceEdit:9678237] Pilco-Janeta, Daniel, 2020年03月13日
schemaClass
Reaction
species
[Species:48887] Homo sapiens
stId
R-HSA-9681382
summation
[Summation:9681377] Ripretinib is a example of a switch pocket inhibitor, a new ...
Referrals
(hasEvent)
[Pathway:R-HSA-9669921] KIT mutants bind TKIs
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