Substituted piperazine

List of substituted piperazines

Benzylpiperazines

Phenylpiperazines

ortho-Substituted

meta-Substituted

para-Substituted

Multiple substitutions

Others

Other arylpiperazines

By drug class

Antianginals

• Ranolazine
• Trimetazidine

Antidepressants

• Amoxapine
• Befuraline
• Buspirone
• Flesinoxan
• Gepirone
• Ipsapirone
• Nefazodone
• Piberaline
• Tandospirone
• Trazodone
• Vilazodone
• Vortioxetine
• Zalospirone

Antihistamines

• Buclizine
• Cetirizine
• Cinnarizine
• Cyclizine
• Hydroxyzine
• Levocetirizine
• Meclizine
• Niaprazine

Antiserotonergics

• EGIS-7625

Antipsychotics

• Typical
  • Flupentixol
  • Fluphenazine
  • Perphenazine
  • Prochlorperazine
  • Thiothixene
  • Trifluoperazine
  • Zuclopenthixol
  • Acetophenazine
  • Carfenazine
• Atypical
  • Amperozide
  • Aripiprazole
  • Clozapine
  • Lurasidone
  • Olanzapine
  • Perospirone
  • Ziprasidone
  • Quetiapine
  • Cariprazine

Recreational Drugs

• 4-Bromo-2,5-dimethoxy-1-benzylpiperazine (2C-B-BZP)
• 1-Benzylpiperazine (BZP)
• 2,3-Dichlorophenylpiperazine (DCPP)
• 1,4-Dibenzylpiperazine (DBZP)
• 4-Methyl-1-benzylpiperazine (MBZP)
• 3-Chlorophenylpiperazine (mCPP)
• 3,4-Methylenedioxy-1-benzylpiperazine (MDBZP)
• 4-Methoxyphenylpiperazine (MeOPP)
• Methoxypiperamide (MeOP or MEXP)
• 4-Chlorophenylpiperazine (pCPP)
• 4-Fluorophenylpiperazine (pFPP)
• 3-Trifluoromethylphenylpiperazine (TFMPP)

Urologicals

• Sildenafil
• Vardenafil

Others

• 6-Nitroquipazine
• Antrafenine
• Diethylcarbamazine
• Diphenazine
• Fipexide
• Imatinib
• NSI-189
• Pipobroman (antineoplastic agent)
• Quipazine
• Sunifiram (nootropic)
• Tolpiprazole (tranquilizer)

Activities

See also

References

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2. ^ Alghamdi, Saad; Alshehri, Mohammed M.; Asif, Mohammad (2022). "The Neuropharmacological Potential of Piperazine Derivatives: A Mini- Review" . Mini-Reviews in Organic Chemistry. 19 (7): 798–810. doi:10.2174/1570193x19666220119120211.
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10. ^ ^{a b c d} Reith ME, Blough BE, Hong WC, Jones KT, Schmitt KC, Baumann MH, Partilla JS, Rothman RB, Katz JL (February 2015). "Behavioral, biological, and chemical perspectives on atypical agents targeting the dopamine transporter". Drug Alcohol Depend. 147: 1–19. doi:10.1016/j.drugalcdep.201412005. PMC 4297708 . PMID 25548026.
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External links