Tetrahydropyridinylpyrrolopyridine

Tetrahydropyridinylpyrrolopyridines are a group of pyrrolopyridine–tetrahydropyridine derivatives related to the tryptamines. They are not tryptamines themselves, as they feature a pyrrolopyridine instead of indole ring system. The compounds include (R)-69, (R)-70, and CP-94253. They are known to act as serotonin receptor agonists, including of the serotonin 5-HT₁ and/or 5-HT₂ receptors.^{[1] [2]} Some tetrahydropyridinylpyrrolopyridines, such as (R)-69 and (R)-70, were discovered by Bryan L. Roth and colleagues via ultra-large-scale docking.^[2]

• Cyclized tryptamine
• Substituted tryptamine § Related compounds
• Indazolethylamine
• Indolizinylethylamine
• List of miscellaneous 5-HT_2A receptor agonists
• Ultra-large-scale docking
• WAY-208466
• Non-hallucinogenic 5-HT_2A receptor agonist