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Schema
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Reaction
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Entries
GRK2 sequesters activated Gq
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authored
[InstanceEdit:416522] Jupe, S, 2009年03月27日 16:14:26
category
binding
compartment
[Compartment:876] plasma membrane
created
[InstanceEdit:416512] Jupe, S, 2009年03月27日 16:11:13
dbId
416516
displayName
GRK2 sequesters activated Gq
edited
[InstanceEdit:435382] Jupe, S, 2009年09月09日
eventOf
[Pathway:R-HSA-416476] G alpha (q) signalling events - Homo sapiens
input
[Complex:R-HSA-114534] G-protein alpha (q/11): GTP [plasma membrane]
[EntityWithAccessionedSequence:R-HSA-50270] GRK2 [plasma membrane]
isInDisease
false
isInferred
false
literatureReference
[LiteratureReference:416514] Selective regulation of Galpha(q/11) by an RGS domain in the G protein-coupled receptor kinase, GRK2
[LiteratureReference:416507] Snapshot of activated G proteins at the membrane: the Galphaq-GRK2-Gbetagamma complex
[LiteratureReference:8983500] Selective regulation of Gq signaling by G protein-coupled receptor kinase 2: direct interaction of kinase N terminus with activated galphaq
maxDepth
1
modified
[InstanceEdit:10867632] Weiser, Joel, 2025年08月27日
name
GRK2 sequesters activated Gq
orthologousEvent
[Reaction:R-HSA-416510] GRK5 sequesters activated Gq - Homo sapiens
[Reaction:R-CEL-416516] GRK2 sequesters activated Gq - Caenorhabditis elegans
[Reaction:R-DME-416516] GRK2 sequesters activated Gq - Drosophila melanogaster
[Reaction:R-GGA-416516] GRK2 sequesters activated Gq - Gallus gallus
[Reaction:R-XTR-416516] GRK2 sequesters activated Gq - Xenopus tropicalis
[Reaction:R-SSC-416516] GRK2 sequesters activated Gq - Sus scrofa
[Reaction:R-BTA-416516] GRK2 sequesters activated Gq - Bos taurus
[Reaction:R-CFA-416516] GRK2 sequesters activated Gq - Canis familiaris
[Reaction:R-RNO-416516] GRK2 sequesters activated Gq - Rattus norvegicus
[Reaction:R-MMU-416516] GRK2 sequesters activated Gq - Mus musculus
output
[Complex:R-HSA-416515] G-protein alpha (q):GRK2 [plasma membrane]
precedingEvent
[Reaction:R-HSA-418576] Dissociation of the P2Y purinoceptor 1:Gq complex - Homo sapiens
[Reaction:R-HSA-397835] Thrombin-activated PARs:Gq (active) dissociate - Homo sapiens
[Reaction:R-HSA-428752] Dissociation of the TP:Gq complex - Homo sapiens
[Reaction:R-HSA-749452] The Ligand:GPCR:Gq complex dissociates - Homo sapiens
releaseDate
2009年09月30日
reviewStatus
[ReviewStatus:9821382] five stars
reviewed
[InstanceEdit:425201] Akkerman, JW, 2009年06月03日
revised
[InstanceEdit:9012014] Varusai, Thawfeek, 2017年07月10日
schemaClass
Reaction
species
[Species:48887] Homo sapiens
stId
R-HSA-416516
summation
[Summation:416505] GRK2 can inhibit GPCR signaling via phosphorylation-independ...
updateTrackers
[UpdateTracker:9781082] Update Tracker - [Reaction:416516] GRK2 sequesters activated Gq - v61:[addLiteratureReference]
[UpdateTracker:9790832] Update Tracker - [Reaction:416516] GRK2 sequesters activated Gq - v32:[add_removeInput]
[UpdateTracker:9790597] Update Tracker - [Reaction:416516] GRK2 sequesters activated Gq - v33:[add_removeInput]
Referrals
(updatedInstance)
[UpdateTracker:9781082] Update Tracker - [Reaction:416516] GRK2 sequesters activated Gq - v61:[addLiteratureReference]
[UpdateTracker:9790832] Update Tracker - [Reaction:416516] GRK2 sequesters activated Gq - v32:[add_removeInput]
[UpdateTracker:9790597] Update Tracker - [Reaction:416516] GRK2 sequesters activated Gq - v33:[add_removeInput]
(hasEvent)
[Pathway:R-HSA-416476] G alpha (q) signalling events
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