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Schema
>
Reaction
>
Entries
AKT inhibitors block AKT membrane recruitment
Show undefined attributes
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authored
[InstanceEdit:2422427] Orlic-Milacic, M, 2012年07月18日
category
binding
compartment
[Compartment:70101] cytosol
created
[InstanceEdit:2400005] Orlic-Milacic, M, 2012年07月13日
crossReference
[DatabaseIdentifier:11944892] Mondo:0004992
dbId
2400010
disease
[Disease:1500689] cancer
displayName
AKT inhibitors block AKT membrane recruitment
edited
[InstanceEdit:2426555] Matthews, L, 2012年08月03日
eventOf
[Pathway:R-HSA-5674400] Constitutive Signaling by AKT1 E17K in Cancer - Homo sapiens
input
[DefinedSet:R-ALL-2399923] AKT inhibitors [cytosol]
[CandidateSet:R-HSA-2400013] AKT/AKT1 E17K mutant [cytosol]
isChimeric
false
isInDisease
true
isInferred
false
literatureReference
[LiteratureReference:2399918] Perifosine, a novel alkylphospholipid, inhibits protein kinase B activation
[LiteratureReference:2404237] First-in-man clinical trial of the oral pan-AKT inhibitor MK-2206 in patients with advanced solid tumors
[LiteratureReference:2404210] The Akt activation inhibitor TCN-P inhibits Akt phosphorylation by binding to the PH domain of Akt and blocking its recruitment to the plasma membrane
[LiteratureReference:2399870] Targeting the phosphoinositide 3-kinase pathway in cancer
maxDepth
1
modified
[InstanceEdit:9830342] Matthews, Lisa, 2023年03月08日
name
AKT inhibitors block AKT membrane recruitment
output
[Complex:R-HSA-2400006] AKT inhibitors:AKT [cytosol]
releaseDate
2012年09月18日
reviewStatus
[ReviewStatus:9821382] five stars
reviewed
[InstanceEdit:2463860] Thorpe, Lauren, 2012年08月13日
[InstanceEdit:2463859] Yuzugullu, Haluk, 2012年08月13日
[InstanceEdit:2463854] Zhao, Jean J, 2012年08月13日
schemaClass
Reaction
species
[Species:48887] Homo sapiens
stId
R-HSA-2400010
summation
[Summation:2404224] AKT inhibitors bind AKT and prevent its association with the...
Referrals
(hasEvent)
[Pathway:R-HSA-5674400] Constitutive Signaling by AKT1 E17K in Cancer
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