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Schema
>
DefinedSet
>
Entries
Overexpressed FGFR2 homodimers [plasma membrane]
Show undefined attributes
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catalystActivities
[CatalystActivity:2029976] protein tyrosine kinase activity of Overexpressed FGFR2 homodimers [plasma membrane]
compartment
[Compartment:876] plasma membrane
componentOf
[Complex:R-HSA-2029966] Overexpressed FGFR2:TKIs [plasma membrane] - Homo sapiens
[Complex:R-HSA-2067714] Overexpressed FGFR2 homodimers:GP369 [plasma membrane] - Homo sapiens
consumedByEvent
[Reaction:R-HSA-2029989] Autocatalytic phosphorylation of overexpressed FGFR2 variants - Homo sapiens
[Reaction:R-HSA-2029992] Tyrosine kinase inhibitors bind to overexpressed FGFR2 variants - Homo sapiens
[Reaction:R-HSA-2067713] GP369 inhibits activation of amplified FGFR2 signaling - Homo sapiens
created
[InstanceEdit:2029962] Rothfels, K, 2012年01月05日
crossReference
[DatabaseIdentifier:11944928] Mondo:0001056
[DatabaseIdentifier:11944895] Mondo:0007254
[DatabaseIdentifier:11944892] Mondo:0004992
dbId
2029963
disease
[Disease:1500689] cancer
[Disease:1500576] breast cancer
[Disease:1500687] stomach cancer
displayName
Overexpressed FGFR2 homodimers [plasma membrane]
hasMember
[Complex:R-HSA-2029921] FGFR2b C3 variant dimer [plasma membrane] - Homo sapiens
[Complex:R-HSA-2029938] Overexpressed FGFR2 dimer [plasma membrane] - Homo sapiens
inDisease
true
literatureReference
[LiteratureReference:2023815] Integrative molecular profiling of triple negative breast cancers identifies amplicon drivers and potential therapeutic targets
[LiteratureReference:2023814] Aberrant receptor internalization and enhanced FRS2-dependent signaling contribute to the transforming activity of the fibroblast growth factor receptor 2 IIIb C3 isoform
[LiteratureReference:2023811] AZD2171 shows potent antitumor activity against gastric cancer over-expressing fibroblast growth factor receptor 2/keratinocyte growth factor receptor
maxDepth
3
modified
[InstanceEdit:2067722] Rothfels, K, 2012年01月25日
name
Overexpressed FGFR2 homodimers
producedByEvent
[Reaction:R-HSA-2029988] Dimerization of overexpressed FGFR2 - Homo sapiens
schemaClass
DefinedSet
species
[Species:48887] Homo sapiens
stId
R-HSA-2029963
Referrals
(hasComponent)
[Complex:R-HSA-2067714] Overexpressed FGFR2 homodimers:GP369 [plasma membrane]
[Complex:R-HSA-2029966] Overexpressed FGFR2:TKIs [plasma membrane]
(input)
[Reaction:R-HSA-2067713] GP369 inhibits activation of amplified FGFR2 signaling
[Reaction:R-HSA-2029989] Autocatalytic phosphorylation of overexpressed FGFR2 variants
[Reaction:R-HSA-2029992] Tyrosine kinase inhibitors bind to overexpressed FGFR2 variants
(physicalEntity)
[CatalystActivity:2029976] protein tyrosine kinase activity of Overexpressed FGFR2 homodimers [plasma membrane]
(output)
[Reaction:R-HSA-2029988] Dimerization of overexpressed FGFR2
(diseaseEntity)
[EntityFunctionalStatus:5654470] gain_of_function of Overexpressed FGFR2 homodimers [plasma membrane]
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